Medicinal Chemistry 3 - Unit 2



Historical background, Nomenclature, Stereochemistry, Structure activity relationship, Chemical degradation classification and important products of the following classes.

  • Macrolide: Erythromycin Clarithromycin, Azithromycin.
  • Miscellaneous: Chloramphenicol\*, Clindamycin.
  • Prodrugs: Basic concepts and application of prodrugs design.
  • Antimalarials: Etiology of malaria. Quinolines: SAR, Quinine sulphate, Chloroquine\*, Amodiaquine, Primaquine phosphate, Pamaquine\*, Quinacrine hydrochloride, Mefloquine. Biguanides and dihydro triazines: Cycloguanil pamoate, Proguanil.
  • Miscellaneous: Pyrimethamine, Artesunete, Artemether, Atovoquone.
Unit 2, Medicinal Chemistry 3, B Pharmacy 6th Sem, Carewell Pharma
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